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5DDB

Menin in complex with MI-319

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue 59Q A 601
ChainResidue
ASER155
ATYR319
AMET322
ATYR323
ADMS602
ADMS607
AHOH761
AHOH807
AHOH982
ALEU177
ASER178
AASP180
AHIS181
AALA182
ATYR276
AMET278
AASN282

site_idAC2
Number of Residues3
Detailsbinding site for residue DMS A 602
ChainResidue
ASER155
A59Q601
ADMS607

site_idAC3
Number of Residues6
Detailsbinding site for residue DMS A 603
ChainResidue
APHE43
APHE47
AGLY386
AGLN400
AHOH793
AHOH955

site_idAC4
Number of Residues6
Detailsbinding site for residue PG4 A 604
ChainResidue
ALEU75
ATHR76
APHE365
AHIS433
AHOH724
AHOH752

site_idAC5
Number of Residues4
Detailsbinding site for residue PG4 A 605
ChainResidue
AGLU274
ALYS304
AHOH723
AHOH778

site_idAC6
Number of Residues3
Detailsbinding site for residue PEG A 606
ChainResidue
ATRP126
ALYS135
ATRP198

site_idAC7
Number of Residues4
Detailsbinding site for residue DMS A 607
ChainResidue
ASER155
APHE238
A59Q601
ADMS602

site_idAC8
Number of Residues4
Detailsbinding site for residue SO4 A 608
ChainResidue
ATYR133
APHE134
AARG137
AARG332

site_idAC9
Number of Residues5
Detailsbinding site for residue SO4 A 609
ChainResidue
AARG108
AGLY111
AGLY169
AARG171
AHOH736

site_idAD1
Number of Residues3
Detailsbinding site for residue SO4 A 610
ChainResidue
ALYS377
AARG446
AHOH808

site_idAD2
Number of Residues2
Detailsbinding site for residue DMS A 611
ChainResidue
AARG207
AGLY294

site_idAD3
Number of Residues5
Detailsbinding site for residue DMS A 612
ChainResidue
AGLY190
AGLU191
ATYR227
AARG229
ASER583

site_idAD4
Number of Residues5
Detailsbinding site for residue SO4 A 613
ChainResidue
AARG332
AVAL334
AARG335
AALA403
AHOH716

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:24275569
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER543

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PDB entries from 2024-07-17

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