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5D3T

First bromodomain of BRD4 bound to inhibitor XD47

Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue 56Y A 201
ChainResidue
ATRP81
ATYR139
AASN140
AHOH305
AHOH312
AHOH320
AHOH397
AHOH398
APRO82
APHE83
AVAL87
ALYS91
ALEU92
ALEU94
AASP96
AILE100

site_idAC2
Number of Residues4
Detailsbinding site for residue NA A 202
ChainResidue
ATYR137
AILE138
AASN140
AGLU163

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO A 203
ChainResidue
AARG58
AGLN59
ALYS102
ATHR103
AHOH328
AHOH425

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

222624

PDB entries from 2024-07-17

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