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5CTB

Humanized yeast ACC carboxyltransferase domain bound to 6,7-dimethyl-1'-[(7-methyl-1H-indazol-5-yl)carbonyl]spiro[chromene-2,4'-piperidin]-4(3H)-one

Functional Information from GO Data
ChainGOidnamespacecontents
A0003989molecular_functionacetyl-CoA carboxylase activity
A0016874molecular_functionligase activity
B0003989molecular_functionacetyl-CoA carboxylase activity
B0016874molecular_functionligase activity
C0003989molecular_functionacetyl-CoA carboxylase activity
C0016874molecular_functionligase activity
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 57J A 2301
ChainResidue
ATHR1757
ALEU2025
AGLU2026
AGLY2029
AGLU2032
AHOH2603
AALA1761
ALYS1764
AVAL1765
AVAL1923
AARG1954
APHE1956
ASER1957
AGLY1958

site_idAC2
Number of Residues4
Detailsbinding site for residue SO4 A 2302
ChainResidue
AARG2154
ASER2157
ATRP2158
ALYS2185

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 2303
ChainResidue
AGLU1750
AGLY1751
ALEU1775
AGLY1779
ATHR1780
AGLN1781

site_idAC4
Number of Residues15
Detailsbinding site for residue 57J B 2301
ChainResidue
BVAL1923
BARG1954
BPHE1956
BGLY1958
BLEU2025
BGLU2026
BGLY2029
BGLU2032
BHOH2435
BHOH2531
CTHR1757
CALA1761
CLEU1762
CLYS1764
CVAL1765

site_idAC5
Number of Residues13
Detailsbinding site for residue 57J C 2301
ChainResidue
BTHR1757
BALA1761
BLEU1762
BLYS1764
BVAL1765
CARG1954
CPHE1956
CGLY1958
CLEU2025
CGLU2026
CGLY2029
CGLU2032
CHOH2503

site_idAC6
Number of Residues5
Detailsbinding site for residue SO4 C 2302
ChainResidue
CARG2125
CARG2128
CHIS2165
CGLU2166
CHOH2465

site_idAC7
Number of Residues4
Detailsbinding site for residue SO4 C 2303
ChainResidue
CARG2154
CTRP2158
CLYS2185
CLEU2189

site_idAC8
Number of Residues6
Detailsbinding site for residue SO4 C 2304
ChainResidue
CGLY1751
CLEU1775
CGLY1779
CTHR1780
CGLN1781
CHOH2666

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues15
DetailsBINDING:
ChainResidueDetails
AALA1627
BARG2036
CALA1627
CARG1731
CGLY1998
CLYS2034
CARG2036
AARG1731
AGLY1998
ALYS2034
AARG2036
BALA1627
BARG1731
BGLY1998
BLYS2034

223166

PDB entries from 2024-07-31

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