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5CCZ

Crystal structure of Mycobacterium tuberculosis malate synthase in complex with 3-(4-fluorophenyl)-4-methyl-1H-pyrazol-5-amine

Functional Information from GO Data
ChainGOidnamespacecontents
A0000287molecular_functionmagnesium ion binding
A0001968molecular_functionfibronectin binding
A0003824molecular_functioncatalytic activity
A0004474molecular_functionmalate synthase activity
A0005515molecular_functionprotein binding
A0005518molecular_functioncollagen binding
A0005576cellular_componentextracellular region
A0005737cellular_componentcytoplasm
A0005829cellular_componentcytosol
A0005886cellular_componentplasma membrane
A0006097biological_processglyoxylate cycle
A0006099biological_processtricarboxylic acid cycle
A0009274cellular_componentpeptidoglycan-based cell wall
A0009436biological_processglyoxylate catabolic process
A0009986cellular_componentcell surface
A0015936biological_processcoenzyme A metabolic process
A0016740molecular_functiontransferase activity
A0042603cellular_componentcapsule
A0042803molecular_functionprotein homodimerization activity
A0043236molecular_functionlaminin binding
A0044406biological_processadhesion of symbiont to host
A0046810molecular_functionhost cell extracellular matrix binding
A0046872molecular_functionmetal ion binding
A0120225molecular_functioncoenzyme A binding
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 50C A 801
ChainResidue
AVAL118
AHOH942
AHOH1026
AHOH1041
AHOH1169
AVAL119
APRO120
ASER275
AMET515
ATRP541
AMET631
AGLU632
AASP633

site_idAC2
Number of Residues6
Detailsbinding site for residue MG A 802
ChainResidue
AGLU434
AASP462
AHOH991
AHOH1042
AHOH1087
AHOH1236

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsActive site: {"description":"Proton acceptor"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsActive site: {"description":"Proton donor"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues18
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues1
DetailsModified residue: {"description":"Cysteine sulfenic acid (-SOH)","evidences":[{"source":"HAMAP-Rule","id":"MF_00641","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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