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5C4O

Identification of a Novel Allosteric Binding Site for RORgt Inhibitors

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 4F1 A 601
ChainResidue
ALEU324
AALA496
AALA497
APHE498
ALEU501
ALEU505
APHE506
ATHR325
AILE328
AGLN329
ALEU353
AMET358
ALEU483
AGLN484
AGLN487

site_idAC2
Number of Residues1
Detailsbinding site for residue GOL A 602
ChainResidue
AHOH703

site_idAC3
Number of Residues2
Detailsbinding site for residue GOL A 603
ChainResidue
AGLN329
AGLU333

site_idAC4
Number of Residues11
Detailsbinding site for residue GOL A 604
ChainResidue
AGLN309
ALYS311
ASER312
AMET313
AARG389
AALA390
ASER413
AASP415
AHIS453
ATHR457
AGOL605

site_idAC5
Number of Residues9
Detailsbinding site for residue GOL A 605
ChainResidue
AARG389
ASER413
AASP415
AGLU416
AHIS453
ALEU454
ATHR457
AARG459
AGOL604

site_idAC6
Number of Residues3
Detailsbinding site for residue SO4 A 606
ChainResidue
AARG302
AGLN309
AARG389

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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