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5C0K

Fragment-Based Drug Discovery Targeting Inhibitor of Apoptosis Proteins: Compound 3

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS300
ACYS303
AHIS320
ACYS327

site_idAC2
Number of Residues12
Detailsbinding site for residue EDO A 402
ChainResidue
ATRP275
AALA291
AGLY293
AEDO403
AEDO403
AHOH501
AHOH506
ATHR271
APHE272
APHE272
AGLY273
ATHR274

site_idAC3
Number of Residues9
Detailsbinding site for residue EDO A 403
ChainResidue
APHE272
ATHR274
ATRP275
ATYR277
AGLY295
AEDO402
AEDO402
AHOH501
AHOH513

site_idAC4
Number of Residues9
Detailsbinding site for residue 4WK A 404
ChainResidue
ALEU307
ATHR308
AASP309
AGLU314
AGLN319
ATRP323
AHOH526
AHOH545
AHOH566

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues66
DetailsBIR_REPEAT_1 BIR repeat. YeaRiftfgt.Wiysvnkeqlar...AGFyAlgegDkvkCfhCgggltdWkpsedpweqHakwyPgCkyL
ChainResidueDetails
ATYR265-LEU330

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00029
ChainResidueDetails
ACYS300
ACYS303
AHIS320
ACYS327

site_idSWS_FT_FI2
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:12747801
ChainResidueDetails
ALYS322
ALYS328

222415

PDB entries from 2024-07-10

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