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5B5B

Crystal structure of VDR-LBD complexed with 2-methylidene-26,27-diphenyl-19-nor-1,25-dihydroxyvitamin D3

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
D0003677molecular_functionDNA binding
D0004879molecular_functionnuclear receptor activity
D0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue AKX A 501
ChainResidue
ATYR143
AASP295
AVAL296
AALA299
AHIS393
AGLN396
ALEU223
AVAL230
ASER233
AARG270
ASER271
ASER274
ATRP282
ACYS284

site_idAC2
Number of Residues15
Detailsbinding site for residue AKX D 501
ChainResidue
DTYR143
DLEU223
DLEU226
DVAL230
DSER233
DARG270
DSER271
DSER274
DTRP282
DCYS284
DASP295
DVAL296
DALA299
DHIS393
DGLN396

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues36
DetailsRegion: {"description":"Interaction with coactivator LXXLL motif","evidences":[{"source":"PubMed","id":"15065852","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues16
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"UniProtKB","id":"P11473","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues12
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"15065852","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1RK3","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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