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5AMF

Crystal structure of the bromodomain of human surface epitope engineered BRD1A in complex with 3D Consortium fragment Ethyl 4,5,6,7- tetrahydro-1H-indazole-5-carboxylate (SGC - Diamond I04-1 fragment screening)

Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE TWL A 1143
ChainResidue
AILE54
AVAL59
ATYR67
ACYS106
ATYR109
AASN110
APHE116
AHOH2083
BMET23

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE NA B 1145
ChainResidue
ALYS108
AHOH2089
AHOH2090
BMET107
BASN110
BTYR117

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AriFaqpvSlkevp..DYLdhIkhpMdfatMrkrleaqg..Yknlhefeedfdl.IidNCmkY
ChainResidueDetails
AALA52-TYR109

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS62
BLYS62

222415

PDB entries from 2024-07-10

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