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5AME

Crystal structure of the bromodomain of human surface epitope engineered BRD1A in complex with 3D Consortium fragment 4-acetyl- piperazin-2-one (SGC - Diamond I04-1 fragment screening)

Functional Information from PDB Data
site_idAC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE PW3 B 1145
ChainResidue
BASN110
BPHE116
BHOH2084

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE NA B 1146
ChainResidue
ALYS108
AHOH2109
AHOH2110
BMET107
BASN110
BTYR117

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AriFaqpvSlkevp..DYLdhIkhpMdfatMrkrleaqg..Yknlhefeedfdl.IidNCmkY
ChainResidueDetails
AALA52-TYR109

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues208
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

240971

PDB entries from 2025-08-27

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