Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE DMS A 201 |
| Chain | Residue |
| A | ILE94 |
| A | PHE114 |
| A | PHE119 |
| A | HOH2126 |
| site_id | AC2 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE DMS A 202 |
| Chain | Residue |
| B | GLY105 |
| B | SER106 |
| A | ARG43 |
| A | HOH2160 |
| B | ALA24 |
| B | LEU25 |
| B | LEU26 |
| site_id | AC3 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE DMS A 203 |
| Chain | Residue |
| A | LEU50 |
| A | TRP60 |
| A | PHE84 |
| A | HOH2159 |
| site_id | AC4 |
| Number of Residues | 3 |
| Details | BINDING SITE FOR RESIDUE DMS A 204 |
| Chain | Residue |
| A | ARG111 |
| A | HOH2026 |
| B | HIS63 |
| site_id | AC5 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO A 300 |
| Chain | Residue |
| A | ALA57 |
| A | ILE58 |
| A | HOH2030 |
| A | HOH2095 |
| B | GLU5 |
| B | LEU9 |
| site_id | AC6 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO A 301 |
| Chain | Residue |
| A | ASP59 |
| A | GLU61 |
| A | THR62 |
| B | EDO301 |
| B | HOH2022 |
| site_id | AC7 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO A 302 |
| Chain | Residue |
| A | ALA57 |
| A | PHE84 |
| A | THR85 |
| A | HOH2095 |
| A | HOH2097 |
| A | HOH2161 |
| B | GLU5 |
| site_id | AC8 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO A 304 |
| Chain | Residue |
| A | LEU17 |
| A | ASP20 |
| A | HOH2035 |
| A | HOH2045 |
| A | HOH2047 |
| site_id | AC9 |
| Number of Residues | 8 |
| Details | BINDING SITE FOR RESIDUE EDO A 305 |
| Chain | Residue |
| A | ALA12 |
| A | ASN15 |
| A | HOH2016 |
| A | HOH2031 |
| B | ALA12 |
| B | ASN15 |
| B | HOH2021 |
| B | HOH2027 |
| site_id | BC1 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO A 306 |
| Chain | Residue |
| A | PRO36 |
| A | MET37 |
| A | LEU116 |
| A | MET120 |
| A | MET123 |
| A | ALA124 |
| A | HOH2162 |
| site_id | BC2 |
| Number of Residues | 9 |
| Details | BINDING SITE FOR RESIDUE EDO A 308 |
| Chain | Residue |
| A | ILE94 |
| A | ARG95 |
| A | PHE114 |
| A | ASP115 |
| A | GLN118 |
| A | HOH2134 |
| A | HOH2135 |
| A | HOH2151 |
| B | VAL35 |
| site_id | BC3 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE DMS B 200 |
| Chain | Residue |
| B | ASP82 |
| B | PHE84 |
| B | ILE94 |
| B | ASP112 |
| site_id | BC4 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE DMS B 204 |
| Chain | Residue |
| A | HIS63 |
| A | GLU79 |
| B | ARG111 |
| B | HOH2138 |
| site_id | BC5 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO B 300 |
| Chain | Residue |
| A | GLU5 |
| A | LEU9 |
| A | HOH2018 |
| B | ALA57 |
| B | ILE58 |
| B | HOH2028 |
| site_id | BC6 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO B 301 |
| Chain | Residue |
| A | EDO301 |
| A | HOH2019 |
| B | ASP59 |
| B | GLU61 |
| B | THR62 |
| site_id | BC7 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO B 302 |
| Chain | Residue |
| A | HOH2018 |
| B | ALA57 |
| B | ASP59 |
| B | PHE84 |
| B | THR85 |
| B | THR91 |
| B | HOH2139 |
| site_id | BC8 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO B 303 |
| Chain | Residue |
| A | ASP20 |
| A | HOH2047 |
| B | ARG13 |
| B | LEU25 |
| B | HOH2140 |
| site_id | BC9 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO B 307 |
| Chain | Residue |
| B | MET1 |
| B | HOH2014 |
| A | ARG47 |
| A | ALA48 |
| A | HOH2080 |
| site_id | CC1 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO B 309 |
| Chain | Residue |
| B | LEU17 |
| B | ASP18 |
| B | LEU19 |
| B | ASP20 |
| B | ARG47 |