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5AEH

Crystal structure of human tankyrase 2 in complex with OD332

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 8IR A 1170
ChainResidue
ASER1033
ATYR1071
AILE1075
APHE1035
AALA1038
AGLY1043
AASP1045
AHIS1048
AGLY1058
AILE1059
ATYR1060

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1173
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC3
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 8IR B 1170
ChainResidue
BSER1033
BPHE1035
BGLY1043
BPHE1044
BASP1045
BHIS1048
BGLY1058
BILE1059
BTYR1060
BTYR1071
BILE1075

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 1173
ChainResidue
BCYS1081
BHIS1084
BCYS1089
BCYS1092

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
BCYS1081
BHIS1084
BCYS1089
BCYS1092

225399

PDB entries from 2024-09-25

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