4ZT6
Trypanosoma brucei methionyl-tRNA synthetase in complex with inhibitor N-[(4R)-6,8-dichloro-3,4-dihydro-2H-chromen-4-yl]-N'-(5-fluoro-1H-imidazo[4,5-b]pyridin-2-yl)propane-1,3-diamine (Chem 1709)
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0000166 | molecular_function | nucleotide binding |
A | 0004812 | molecular_function | aminoacyl-tRNA ligase activity |
A | 0004825 | molecular_function | methionine-tRNA ligase activity |
A | 0005524 | molecular_function | ATP binding |
A | 0006418 | biological_process | tRNA aminoacylation for protein translation |
A | 0006431 | biological_process | methionyl-tRNA aminoacylation |
B | 0000166 | molecular_function | nucleotide binding |
B | 0004812 | molecular_function | aminoacyl-tRNA ligase activity |
B | 0004825 | molecular_function | methionine-tRNA ligase activity |
B | 0005524 | molecular_function | ATP binding |
B | 0006418 | biological_process | tRNA aminoacylation for protein translation |
B | 0006431 | biological_process | methionyl-tRNA aminoacylation |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 8 |
Details | binding site for residue MET A 801 |
Chain | Residue |
A | ILE248 |
A | TYR250 |
A | ASP287 |
A | TRP474 |
A | TYR481 |
A | HIS523 |
A | HOH933 |
A | HOH986 |
site_id | AC2 |
Number of Residues | 2 |
Details | binding site for residue DMS A 802 |
Chain | Residue |
A | DMS803 |
A | LYS521 |
site_id | AC3 |
Number of Residues | 4 |
Details | binding site for residue DMS A 803 |
Chain | Residue |
A | GLU392 |
A | ASP518 |
A | LYS521 |
A | DMS802 |
site_id | AC4 |
Number of Residues | 4 |
Details | binding site for residue DMS A 804 |
Chain | Residue |
A | TRP345 |
A | GLU349 |
A | VAL463 |
A | PRO464 |
site_id | AC5 |
Number of Residues | 3 |
Details | binding site for residue DMS B 801 |
Chain | Residue |
B | TYR324 |
B | SER325 |
B | ILE326 |
site_id | AC6 |
Number of Residues | 18 |
Details | binding site for residue 4RD B 802 |
Chain | Residue |
B | PRO247 |
B | ILE248 |
B | TYR250 |
B | ASP287 |
B | GLY290 |
B | LEU456 |
B | VAL471 |
B | TYR472 |
B | VAL473 |
B | TRP474 |
B | ASP476 |
B | TYR481 |
B | ILE519 |
B | PHE522 |
B | HIS523 |
B | HOH940 |
B | HOH946 |
B | HOH950 |