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4ZNH

Crystal Structure of the ER-alpha Ligand-binding Domain (Y537S) in complex with a 2-Fluoro-substituted OBHS derivative

Functional Information from PDB Data
site_idAC1
Number of Residues21
Detailsbinding site for residue OBC A 601
ChainResidue
AMET343
AVAL418
AGLU419
AGLY420
AMET421
AILE424
AGLY521
AHIS524
ALEU525
AMET528
ALEU540
ALEU346
AOBC602
AHOH748
ATHR347
AALA350
AGLU353
ALEU387
AMET388
AARG394
APHE404

site_idAC2
Number of Residues19
Detailsbinding site for residue OBC A 602
ChainResidue
AMET343
ATHR347
AALA350
AGLU353
ALEU387
AMET388
AARG394
APHE404
AVAL418
AGLU419
AGLY420
AMET421
AILE424
AGLY521
AHIS524
ALEU525
ALEU540
AOBC601
AHOH748

site_idAC3
Number of Residues19
Detailsbinding site for residue OBC B 601
ChainResidue
BMET343
BTHR347
BALA350
BGLU353
BLEU387
BMET388
BARG394
BPHE404
BVAL418
BGLU419
BGLY420
BMET421
BILE424
BGLY521
BHIS524
BLEU525
BMET528
BLEU540
BHOH734

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ASER537
BSER537

site_idSWS_FT_FI2
Number of Residues2
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
BCYS447

222624

PDB entries from 2024-07-17

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