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4YPA

ASH1L SET domain Q2265A mutant in complex with S-adenosyl methionine (SAM)

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0042054molecular_functionhistone methyltransferase activity
B0005634cellular_componentnucleus
B0042054molecular_functionhistone methyltransferase activity
C0005634cellular_componentnucleus
C0042054molecular_functionhistone methyltransferase activity
D0005634cellular_componentnucleus
D0042054molecular_functionhistone methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 3001
ChainResidue
ACYS2091
ACYS2093
ACYS2104
ACYS2108

site_idAC2
Number of Residues4
Detailsbinding site for residue ZN A 3002
ChainResidue
ACYS2104
ACYS2117
ACYS2122
ACYS2128

site_idAC3
Number of Residues4
Detailsbinding site for residue ZN A 3003
ChainResidue
ACYS2268
ACYS2270
ACYS2275
ACYS2220

site_idAC4
Number of Residues18
Detailsbinding site for residue SAM A 3004
ChainResidue
ALYS2150
ATRP2152
ASER2191
AASP2192
AHIS2193
ATYR2194
AARG2214
APHE2215
AILE2216
AASN2217
AHIS2218
ATYR2255
AGLN2266
ALEU2267
ACYS2268
ALYS2269
AILE2279
AHOH3131

site_idAC5
Number of Residues4
Detailsbinding site for residue ZN B 2301
ChainResidue
BCYS2091
BCYS2093
BCYS2104
BCYS2108

site_idAC6
Number of Residues4
Detailsbinding site for residue ZN B 2302
ChainResidue
BCYS2104
BCYS2117
BCYS2122
BCYS2128

site_idAC7
Number of Residues4
Detailsbinding site for residue ZN B 2303
ChainResidue
BCYS2220
BCYS2268
BCYS2270
BCYS2275

site_idAC8
Number of Residues13
Detailsbinding site for residue SAM B 2304
ChainResidue
BLYS2150
BTRP2152
BASP2192
BHIS2193
BTYR2194
BARG2214
BASN2217
BHIS2218
BTYR2255
BGLN2266
BLEU2267
BLYS2269
BILE2279

site_idAC9
Number of Residues4
Detailsbinding site for residue ZN C 2301
ChainResidue
CCYS2091
CCYS2093
CCYS2104
CCYS2108

site_idAD1
Number of Residues4
Detailsbinding site for residue ZN C 2302
ChainResidue
CCYS2104
CCYS2117
CCYS2122
CCYS2128

site_idAD2
Number of Residues4
Detailsbinding site for residue ZN C 2303
ChainResidue
CCYS2220
CCYS2268
CCYS2270
CCYS2275

site_idAD3
Number of Residues16
Detailsbinding site for residue SAM C 2304
ChainResidue
CLYS2150
CTRP2152
CSER2191
CASP2192
CHIS2193
CTYR2194
CARG2214
CPHE2215
CASN2217
CHIS2218
CTYR2255
CGLN2266
CLEU2267
CCYS2268
CLYS2269
CILE2279

site_idAD4
Number of Residues5
Detailsbinding site for residue ZN D 2301
ChainResidue
DCYS2091
DCYS2093
DCYS2104
DCYS2108
DZN2302

site_idAD5
Number of Residues5
Detailsbinding site for residue ZN D 2302
ChainResidue
DCYS2104
DCYS2117
DCYS2122
DCYS2128
DZN2301

site_idAD6
Number of Residues4
Detailsbinding site for residue ZN D 2303
ChainResidue
DCYS2220
DCYS2268
DCYS2270
DCYS2275

site_idAD7
Number of Residues16
Detailsbinding site for residue SAM D 2304
ChainResidue
DTRP2152
DASP2192
DHIS2193
DTYR2194
DARG2214
DASN2217
DHIS2218
DTYR2255
DGLN2266
DLEU2267
DCYS2268
DLYS2269
DILE2279
DHOH2419
DLYS2150
DGLY2151

219869

PDB entries from 2024-05-15

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