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4X5Y

Menin in complex with MI-503

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
Functional Information from PDB Data
site_idAC1
Number of Residues20
Detailsbinding site for residue 3XW A 601
ChainResidue
ASER155
AMET322
ATYR323
ATRP341
AGLU363
AGLU366
AVAL371
ADMS602
AHOH806
AHOH822
AHOH823
ALEU177
AHOH948
ASER178
AASP180
AHIS181
AALA182
APHE238
ATYR276
AMET278

site_idAC2
Number of Residues3
Detailsbinding site for residue DMS A 602
ChainResidue
A3XW601
AHOH827
AHOH828

site_idAC3
Number of Residues8
Detailsbinding site for residue PG4 A 603
ChainResidue
ALEU75
ATHR76
ATYR361
APHE365
AHOH708
AHOH711
AHOH870
AHOH1009

site_idAC4
Number of Residues3
Detailsbinding site for residue SO4 A 604
ChainResidue
APRO12
AARG14
AHOH973

site_idAC5
Number of Residues4
Detailsbinding site for residue SO4 A 605
ChainResidue
ATYR133
APHE134
AARG137
AARG332

site_idAC6
Number of Residues2
Detailsbinding site for residue SO4 A 606
ChainResidue
ALYS377
AARG446

site_idAC7
Number of Residues5
Detailsbinding site for residue DMS A 607
ChainResidue
APHE43
APHE47
AGLN400
AHOH885
AHOH895

site_idAC8
Number of Residues6
Detailsbinding site for residue DMS A 608
ChainResidue
AVAL185
AGLY190
AGLU191
ATYR227
AARG229
ASER583

site_idAC9
Number of Residues2
Detailsbinding site for residue 04E A 609
ChainResidue
ATRP126
ALYS135

site_idAD1
Number of Residues7
Detailsbinding site for residue EPE A 610
ChainResidue
AVAL50
AASN331
AARG332
AVAL334
AARG335
AGLY401
AALA403

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER543

225158

PDB entries from 2024-09-18

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