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4WH8

Crystal Structure of HCV NS3/4A protease in complex with an Asunaprevir P1-P3 macrocyclic analog.

Functional Information from GO Data
ChainGOidnamespacecontents
A0006508biological_processproteolysis
A0008236molecular_functionserine-type peptidase activity
A0019087biological_processtransformation of host cell by virus
B0006508biological_processproteolysis
B0008236molecular_functionserine-type peptidase activity
B0019087biological_processtransformation of host cell by virus
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 3M7 A 1201
ChainResidue
AGLN1041
ASER1138
AALA1139
APHE1154
AARG1155
AALA1156
AALA1157
APHE1043
AHIS1057
AGLY1058
AVAL1078
AASP1081
ALEU1135
ALYS1136
AGLY1137

site_idAC2
Number of Residues5
Detailsbinding site for residue SO4 A 1202
ChainResidue
ATYR1006
AGLN1008
AHOH1302
AHOH1306
BTYR1056

site_idAC3
Number of Residues5
Detailsbinding site for residue SO4 A 1203
ChainResidue
ATYR1056
AHOH1314
AHOH1317
BTYR1006
BGLN1008

site_idAC4
Number of Residues4
Detailsbinding site for residue ZN A 1204
ChainResidue
ACYS1097
ACYS1099
ACYS1145
AHIS1149

site_idAC5
Number of Residues14
Detailsbinding site for residue 3M7 B 1201
ChainResidue
BGLN1041
BPHE1043
BHIS1057
BVAL1078
BASP1081
BLEU1135
BLYS1136
BGLY1137
BSER1138
BALA1139
BPHE1154
BARG1155
BALA1156
BALA1157

site_idAC6
Number of Residues4
Detailsbinding site for residue ZN B 1202
ChainResidue
BCYS1097
BCYS1099
BCYS1145
BHIS1149

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PDB entries from 2024-07-31

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