4W9Q
The Fk1 domain of FKBP51 in complex with (1S,5S,6R)-10-[(3,5-dichlorophenyl)sulfonyl]-3-[2-(3,4-dimethoxyphenoxy)ethyl]-5-ethyl-3,10-diazabicyclo[4.3.1]decan-2-one
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003755 | molecular_function | peptidyl-prolyl cis-trans isomerase activity |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 17 |
Details | binding site for residue 3JP A 201 |
Chain | Residue |
A | TYR57 |
A | TYR113 |
A | SER118 |
A | LYS121 |
A | PHE130 |
A | HOH359 |
A | HOH502 |
A | HOH516 |
A | HOH518 |
A | PHE67 |
A | ASP68 |
A | GLY84 |
A | GLN85 |
A | VAL86 |
A | ILE87 |
A | TRP90 |
A | ALA112 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | MOD_RES: N6-acetyllysine => ECO:0000269|PubMed:28147277 |
Chain | Residue | Details |
A | LYS28 |