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4W9Q

The Fk1 domain of FKBP51 in complex with (1S,5S,6R)-10-[(3,5-dichlorophenyl)sulfonyl]-3-[2-(3,4-dimethoxyphenoxy)ethyl]-5-ethyl-3,10-diazabicyclo[4.3.1]decan-2-one

Functional Information from GO Data
ChainGOidnamespacecontents
A0003755molecular_functionpeptidyl-prolyl cis-trans isomerase activity
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue 3JP A 201
ChainResidue
ATYR57
ATYR113
ASER118
ALYS121
APHE130
AHOH359
AHOH502
AHOH516
AHOH518
APHE67
AASP68
AGLY84
AGLN85
AVAL86
AILE87
ATRP90
AALA112

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000269|PubMed:28147277
ChainResidueDetails
ALYS28

225681

PDB entries from 2024-10-02

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