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4UXH

Leishmania major Thymidine Kinase in complex with AP5dT

Functional Information from GO Data
ChainGOidnamespacecontents
A0004797molecular_functionthymidine kinase activity
A0005524molecular_functionATP binding
B0004797molecular_functionthymidine kinase activity
B0005524molecular_functionATP binding
Functional Information from PDB Data
site_idAC1
Number of Residues36
DetailsBINDING SITE FOR RESIDUE T5A A 1180
ChainResidue
AMET13
AASP43
AARG45
ATYR46
AGLU85
AGLN87
APHE88
ALEU111
AASP114
ATYR115
APHE120
APHE14
ATHR151
AARG153
AGLN160
AGLU161
ALEU162
AILE163
AGLY164
ATYR169
AHOH2002
AHOH2003
AALA15
AHOH2005
AHOH2006
AHOH2007
AHOH2012
AHOH2013
AHOH2035
BHIS30
AGLY16
ALYS17
ATHR18
ATHR19
AMET22
ALYS39

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1181
ChainResidue
ACYS140
ACYS143
ACYS173
ACYS176

site_idAC3
Number of Residues30
DetailsBINDING SITE FOR RESIDUE T5A B 1182
ChainResidue
AHIS30
BMET13
BPHE14
BALA15
BGLY16
BLYS17
BTHR18
BTHR19
BMET22
BLYS39
BASP43
BGLU85
BGLN87
BPHE88
BLEU111
BASP114
BTYR115
BPHE120
BARG153
BGLN160
BGLU161
BLEU162
BILE163
BGLY164
BTYR169
BHOH2002
BHOH2003
BHOH2005
BHOH2006
BHOH2022

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 1183
ChainResidue
BCYS140
BCYS143
BCYS173
BCYS176

Functional Information from PROSITE/UniProt
site_idPS00603
Number of Residues14
DetailsTK_CELLULAR_TYPE Thymidine kinase cellular-type signature. GgaDmYiAtCReCY
ChainResidueDetails
AGLY164-TYR177

224572

PDB entries from 2024-09-04

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