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4UVZ

Crystal structure of human tankyrase 2 in complex with 5-amino-3- phenyl-1,2-dihydroisoquinolin-1-one

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2162
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN C 2162
ChainResidue
CCYS1081
CHIS1084
CCYS1089
CCYS1092

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 2163
ChainResidue
AHIS979
AARG980
ALYS1067
AHOH3046
AHOH3178
AHOH3261
AARG977

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 C 2163
ChainResidue
CARG977
CHIS979
CARG980
CLYS1067
CGLN1070

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 2164
ChainResidue
AASN990
AARG991
APRO1160
AGLU1161
AHOH3070
AHOH3072

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 C 2164
ChainResidue
CASN990
CARG991
CPRO1160
CGLU1161
CHOH3062
CHOH3065
CHOH3219

site_idAC7
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 5NN C 2165
ChainResidue
CHIS1031
CGLY1032
CTYR1050
CTYR1060
CALA1062
CLYS1067
CSER1068
CTYR1071
CGLU1138

site_idAC8
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 5NN A 2165
ChainResidue
AHIS1031
AGLY1032
ATYR1050
ATYR1060
AALA1062
ALYS1067
ASER1068
ATYR1071
AGLU1138

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 2166
ChainResidue
APRO1129
ASER1130
AVAL1131
AASN1132
AGLY1133

site_idBC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE PEG C 2166
ChainResidue
CTYR1148
CGLU1150

site_idBC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE PEG A 2167
ChainResidue
AASN1002
ATRP1006
ATYR1148
AGLU1150

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
CCYS1081
CHIS1084
CCYS1089
CCYS1092

222415

PDB entries from 2024-07-10

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