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4UUG

The (R)-selective amine transaminase from Aspergillus fumigatus with inhibitor bound

Functional Information from GO Data
ChainGOidnamespacecontents
A0003824molecular_functioncatalytic activity
A0005575cellular_componentcellular_component
A0008483molecular_functiontransaminase activity
A0019752biological_processcarboxylic acid metabolic process
A0046394biological_processcarboxylic acid biosynthetic process
B0003824molecular_functioncatalytic activity
B0005575cellular_componentcellular_component
B0008483molecular_functiontransaminase activity
B0019752biological_processcarboxylic acid metabolic process
B0046394biological_processcarboxylic acid biosynthetic process
Functional Information from PDB Data
site_idAC1
Number of Residues23
DetailsBINDING SITE FOR RESIDUE PXG A 401
ChainResidue
ATYR58
AASN217
ALEU234
AGLY236
AILE237
ATHR238
ATHR273
ATHR274
AALA275
AMRD402
AHOH2111
AARG77
AHOH2112
AHOH2113
AHOH2304
BHIS53
APHE113
ALYS179
ATRP183
AGLU212
AGLY213
AGLY215
APHE216

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE MRD A 402
ChainResidue
APHE113
ALEU143
APXG401
AHOH2185
AHOH2415
BMET52
BHIS53
BVAL125

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE FMT A 403
ChainResidue
ASER62
ATYR145
ATHR274
ATYR305
ATRP306
AHIS309

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE FMT A 404
ChainResidue
AARG164
AHOH2285
AHOH2416

site_idAC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE FMT A 405
ChainResidue
AMET85
AARG120
AHOH2187
AHOH2418
AHOH2419
BLYS188
BPHE191

site_idAC6
Number of Residues23
DetailsBINDING SITE FOR RESIDUE PXG B 401
ChainResidue
AHOH2103
AHOH2196
AHOH2198
BTYR58
BARG77
BPHE113
BLYS179
BTRP183
BGLU212
BGLY213
BGLY215
BPHE216
BASN217
BLEU234
BGLY236
BILE237
BTHR238
BTHR273
BTHR274
BALA275
BHOH2085
BHOH2086
BHOH2268

site_idAC7
Number of Residues8
DetailsBINDING SITE FOR RESIDUE MPD B 402
ChainResidue
ALEU47
AHIS53
AHOH2073
AHOH2092
AHOH2190
BPHE113
BLEU143
BHOH2375

site_idAC8
Number of Residues6
DetailsBINDING SITE FOR RESIDUE FMT B 403
ChainResidue
BSER62
BTYR145
BTHR274
BTYR305
BHIS309
BHOH2089

site_idAC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE FMT B 404
ChainResidue
BARG164
BHOH2246
BHOH2376
BHOH2377

site_idBC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE FMT B 405
ChainResidue
ALEU36
BTYR31
BILE138
BHOH2055
BHOH2182
BHOH2191

site_idBC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE NA B 406
ChainResidue
BHOH2191
BLEU133
BASN136
BASN137
BHOH2181
BHOH2182

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PDB entries from 2024-06-26

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