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4UIZ

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH 7-(3,4-dimethoxyphenyl)-2-(4-methanesulfonylpiperazine-1-carbonyl)-5-methyl-4H,5H-thieno-3,2-c- pyridin-4-one

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1169
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH2190
AHOH2279

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1170
ChainResidue
AN1D1171
AHOH2186
AHOH2281
ALYS99
AILE146

site_idAC3
Number of Residues20
DetailsBINDING SITE FOR RESIDUE N1D A 1171
ChainResidue
ATRP81
APRO82
AGLN85
ALEU92
ALEU94
AASP96
ALYS99
ATYR139
AASN140
AEDO1170
AHOH2093
AHOH2139
AHOH2143
AHOH2169
AHOH2170
AHOH2179
AHOH2180
AHOH2282
AHOH2283
AHOH2284

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

223790

PDB entries from 2024-08-14

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