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4UIY

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH N-(1,1-dioxo-1-thian-4-yl)- 5-methyl-4-oxo-7-3-(trifluoromethyl)phenyl-4H,5H-thieno-3,2-c- pyridine-2-carboximidamide

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1169
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH2169

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1170
ChainResidue
A5V21172
AHOH2144
AHOH2261
AHOH2262
ATRP81
AGLN85
AASP96

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1171
ChainResidue
APRO53
ALYS99
AMET149
A5V21172
AHOH2224
AHOH2263

site_idAC4
Number of Residues16
DetailsBINDING SITE FOR RESIDUE 5V2 A 1172
ChainResidue
ATRP81
APRO82
AVAL87
ALEU92
ALEU94
AASP96
ALYS99
ATYR139
AASN140
ALYS141
AASP144
AEDO1170
AEDO1171
AHOH2147
AHOH2159
AHOH2264

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

218500

PDB entries from 2024-04-17

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