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4UIU

BROMODOMAIN OF HUMAN BRD9 WITH 7-(3,4-dimethoxyphenyl)-N-(1,1-dioxo-1- thian-4-yl)-5-methyl-4-oxo-4H,5H-thieno-3,2-c-pyridine-2-carboxamide

Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE TVU A 1123
ChainResidue
AGLY43
ATYR106
ATYR107
ALYS111
AHOH2115
AHOH2236
AHOH2237
APHE44
APHE45
AVAL49
AILE53
ATYR99
AASN100
AARG101
ATHR104

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding => ECO:0000269|PubMed:26365797
ChainResidueDetails
AILE53
ATYR106

237992

PDB entries from 2025-06-25

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