4UIT
BROMODOMAIN OF HUMAN BRD9 WITH 7-(3,4-dimethoxyphenyl)-2-(4- methanesulfonylpiperazine-1-carbonyl)-5-methyl-4H,5H-thieno-3,2-c- pyridin-4-one
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 16 |
Details | BINDING SITE FOR RESIDUE N1D A 1123 |
Chain | Residue |
A | PHE44 |
A | HOH2067 |
A | HOH2074 |
A | HOH2107 |
A | HOH2185 |
A | HOH2196 |
A | HOH2204 |
A | HOH2205 |
A | PHE45 |
A | ILE53 |
A | ALA54 |
A | TYR99 |
A | ASN100 |
A | ARG101 |
A | TYR106 |
A | LYS111 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | SITE: Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding => ECO:0000269|PubMed:26365797 |
Chain | Residue | Details |
A | ILE53 | |
A | TYR106 |