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4UI7

Crystal structure of human tankyrase 2 in complex with TA-49

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
D0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 2114
ChainResidue
BCYS1081
BHIS1084
BCYS1089
BCYS1092

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2113
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC3
Number of Residues9
DetailsBINDING SITE FOR RESIDUE SO4 A 2114
ChainResidue
AHIS979
AARG980
ALYS1067
AHOH3044
AHOH3051
AHOH3053
AHOH3154
AHOH3155
AARG977

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 2115
ChainResidue
BARG977
BHIS979
BARG980
BLYS1067
BHOH3043
BHOH3126

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 2116
ChainResidue
BASN990
BARG991
BHOH3059
BHOH3063
BHOH3175
DGLU1161

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 2115
ChainResidue
AASN990
AARG991
AHOH3070
AHOH3072
CPRO1160
CGLU1161

site_idAC7
Number of Residues9
DetailsBINDING SITE FOR RESIDUE VT3 A 2116
ChainResidue
AHIS1031
AGLY1032
ASER1033
ATYR1050
ATYR1060
ALYS1067
ASER1068
ATYR1071
CGLU1138

site_idAC8
Number of Residues9
DetailsBINDING SITE FOR RESIDUE VT3 B 2117
ChainResidue
BHIS1031
BGLY1032
BSER1033
BTYR1050
BTYR1060
BLYS1067
BSER1068
BTYR1071
DGLU1138

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL C 2162
ChainResidue
CPRO1129
CSER1130
CVAL1131
CASN1132
CGLY1133

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"O95271","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

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PDB entries from 2025-10-08

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