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4UI3

Crystal structure of human tankyrase 2 in complex with TA-26

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ ADP-ribosyltransferase activity
D0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 2114
ChainResidue
BCYS1081
BHIS1084
BCYS1089
BCYS1092

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2113
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 2115
ChainResidue
BHIS979
BARG980
BLYS1067
BGLN1070
BHOH3034
BHOH3039
BARG977

site_idAC4
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 2114
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070
AHOH3038
AHOH3043
AHOH3125

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 D 2162
ChainResidue
BASN990
BARG991
BHOH3050
DPRO1160
DGLU1161

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 C 2162
ChainResidue
AASN990
AARG991
AHOH3057
AHOH3060
CPRO1160
CGLU1161
CHOH3018

site_idAC7
Number of Residues14
DetailsBINDING SITE FOR RESIDUE 06R A 2115
ChainResidue
AHIS1031
AGLY1032
APRO1034
APHE1035
AALA1049
ATYR1050
ATYR1060
AALA1062
ALYS1067
ASER1068
ATYR1071
AILE1075
AHOH3112
CGLU1138

site_idAC8
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 06R B 2116
ChainResidue
BHIS1031
BGLY1032
BSER1033
BPRO1034
BPHE1035
BALA1049
BTYR1050
BTYR1060
BALA1062
BLYS1067
BSER1068
BTYR1071
DGLU1138

site_idAC9
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL C 2163
ChainResidue
CARG1128
CPRO1129
CSER1130
CVAL1131
CASN1132
CGLY1133
CHOH3012

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
BCYS1081
BHIS1084
BCYS1089
BCYS1092

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PDB entries from 2024-07-17

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