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4TU4

Crystal structure of ATAD2A bromodomain complexed with 3-(3,5-dimethyl-1,2-oxazol-4-yl)-5-[(phenylsulfonyl)amino]benzoicacid

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue SO4 A 1201
ChainResidue
AARG987
AARG990
AARG994
AARG1067
AARG1072
AHOH1342

site_idAC2
Number of Residues6
Detailsbinding site for residue GOL A 1202
ChainResidue
AASP1094
AHOH1315
AHOH1332
AGLU988
AGLU1092
ALEU1093

site_idAC3
Number of Residues3
Detailsbinding site for residue GOL A 1203
ChainResidue
AARG1082
AASP1083
AHOH1385

site_idAC4
Number of Residues9
Detailsbinding site for residue 37N A 1204
ChainResidue
AARG1007
AVAL1008
AVAL1013
AASP1014
AGLU1017
AASN1064
AILE1074
AHOH1366
AHOH1376

site_idAC5
Number of Residues3
Detailsbinding site for residue CL A 1205
ChainResidue
AARG1077
AHOH1325
AHOH1344

site_idAC6
Number of Residues4
Detailsbinding site for residue DMS A 1206
ChainResidue
AVAL1046
ALYS1047
AHOH1419
AHOH1445

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PDB entries from 2024-08-28

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