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4TQN

Crystal structure of the bromodomain of human CREBBP in complex with UL04

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue UL4 A 1201
ChainResidue
ALEU1109
AHOH1335
AHOH1355
APRO1110
AVAL1115
ALEU1120
AASN1168
AARG1173
AVAL1174
AEDO1202
AEDO1203

site_idAC2
Number of Residues2
Detailsbinding site for residue EDO A 1202
ChainResidue
AGLY1121
AUL41201

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 1203
ChainResidue
ALEU1120
AUL41201
AHOH1322
AHOH1327

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 1204
ChainResidue
AILE1128
AVAL1129
ALYS1130
AASN1131
AASN1163

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

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PDB entries from 2024-07-17

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