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4RUO

Crystal structure of zVDR L337H mutant-gemini complex

Functional Information from GO Data
ChainGOidnamespacecontents
X0003677molecular_functionDNA binding
X0004879molecular_functionnuclear receptor activity
X0005634cellular_componentnucleus
X0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE BIV X 501
ChainResidue
XTYR175
XHIS333
XLEU338
XLEU341
XLEU419
XHIS423
XSER265
XILE299
XARG302
XSER303
XSER306
XTRP314
XCYS316
XVAL328

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues18
DetailsRegion: {"description":"Interaction with coactivator LXXLL motif","evidences":[{"source":"UniProtKB","id":"P13053","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"UniProtKB","id":"P11473","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"17218092","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2HC4","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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