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4QST

Structure of the bromodomain of human ATPase family AAA domain-containing protein 2 (ATAD2) in complex with 1-methylquinolin 2-one

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE 12Q A 1201
ChainResidue
AVAL1008
AVAL1013
AVAL1018
AASN1064
AILE1074
AHOH1394
AHOH1397

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1202
ChainResidue
AARG994
AARG1067
AARG1072
AHOH1412
AHOH1443
AARG987
AARG990

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1203
ChainResidue
ALYS1042
ALYS1042
AHOH1373
AHOH1438
AHOH1438
AHOH1458
AHOH1458

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1204
ChainResidue
AGLU988
ALEU1093
AASP1094
APHE1097
AHOH1323
AHOH1352

site_idAC5
Number of Residues8
DetailsBINDING SITE FOR RESIDUE EDO A 1205
ChainResidue
AMET980
AGLU983
AASP984
AARG987
AARG990
AHOH1312
AHOH1442
AHOH1443

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1206
ChainResidue
ALYS1004
AEDO1216
AHOH1314
AHOH1375

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1207
ChainResidue
AILE1089
ALYS1090
ALEU1093
AHOH1377
AHOH1427

site_idAC8
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1208
ChainResidue
AHIS998
AALA1001
AHOH1472

site_idAC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1209
ChainResidue
APRO1012
ASER1032
ASER1033
ASER1036
AHOH1369
AHOH1434

site_idBC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1210
ChainResidue
AHIS998
AGLU1092
AHOH1358
AHOH1427

site_idBC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 1211
ChainResidue
AASP1039
ALEU1040

site_idBC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1212
ChainResidue
APRO1065
AASP1066
AARG1067
AARG1072
AARG1075
AHOH1449

site_idBC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1213
ChainResidue
AGLN981
AGLU982
ATHR985
AARG1072
AHIS1076
AHOH1380
AHOH1426

site_idBC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1214
ChainResidue
AARG990
AHIS1041
ALEU1044
AARG1108
AHOH1374

site_idBC6
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1215
ChainResidue
AASP1054
ACYS1057
ALEU1061
AARG1082
AHOH1418

site_idBC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1216
ChainResidue
AARG1077
AEDO1206
AHOH1311
AHOH1316
AHOH1395

site_idBC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1217
ChainResidue
AARG1082
AASP1083
ATYR1086
AHOH1325
AHOH1422

site_idBC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1218
ChainResidue
APRO1028
ASER1033
AHOH1372
AHOH1402
AHOH1477
AHOH1478

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PDB entries from 2024-04-24

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