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4QC3

Crystal structure of human BAZ2B bromodomain in complex with a diacetylated histone 4 peptide (H4K8acK12ac)

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 2201
ChainResidue
APRO2084
ALEU2087
APRO2088
AHOH2317
AHOH2329
AHOH2375
AHOH2411

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2202
ChainResidue
BLYS2064
AASP2065
ALEU2122

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO B 2201
ChainResidue
AGLY2096
BPHE2139
CALY8
CGLY9

site_idAC4
Number of Residues21
DetailsBINDING SITE FOR CHAIN C OF DIACETYLATED HISTONE 4 PEPTIDE (H4K8ACK12AC)
ChainResidue
APRO2084
AVAL2089
ATHR2138
APHE2139
AASN2140
AILE2146
AHOH2310
AHOH2312
BPRO2084
BVAL2089
BVAL2094
BPRO2095
BASN2140
BILE2146
BEDO2201
BHOH2317
CHOH102
CHOH107
CHOH108
CHOH109
CHOH110

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA2082-PHE2139

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PDB entries from 2024-07-24

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