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4O0J

HIV-1 Integrase Catalytic Core Domain Complexed with Allosteric Inhibitor (2S)-tert-butoxy[4-(4-chlorophenyl)-6-(3,4-dimethylphenyl)-2,5-dimethylpyridin-3-yl]ethanoic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE LF8 A 301
ChainResidue
ATHR124
ATHR174
AHOH406
AHOH452
ATHR125
AALA128
AALA129
ATRP132
AILE141
AALA169
AGLU170
AHIS171

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 302
ChainResidue
AGLY94
AGLN95
ASER123
ATHR124
ATHR125
ALYS186
AHOH407
AHOH409

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 303
ChainResidue
ALYS71
AHIS171
ALEU172
AHOH411
AHOH426

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 304
ChainResidue
ATHR66
AHIS67
ALYS159

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P04585","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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