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4NR7

Crystal structure of the bromodomain of human CREBBP in complex with an isoxazolyl-benzimidazole ligand

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1201
ChainResidue
AARG1091
AMET1095
APRO1096
AASP1124
AHOH1316
AHOH1348

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1202
ChainResidue
ALYS1141
AGLN1146
AHOH1318

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1203
ChainResidue
AGLU1107
AASN1162
ATRP1165
ALEU1166
AHOH1371
AHOH1401
AHOH1469

site_idAC4
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 2LO A 1204
ChainResidue
ALEU1109
APRO1110
AVAL1115
ALEU1120
AILE1122
ATYR1125
AASN1168
AARG1173
AVAL1174
APHE1177
AHOH1306
AHOH1498
AHOH1501

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

221716

PDB entries from 2024-06-26

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