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4NR5

Crystal structure of the bromodomain of human CREBBP in complex with an isoxazolyl-benzimidazole ligand

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 2LL A 1201
ChainResidue
APRO1110
ATYR1175
ANO31202
AEDO1203
AHOH1309
AVAL1115
ALEU1119
ALEU1120
ATRP1158
ATRP1165
AASN1168
ALYS1170
AVAL1174

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE NO3 A 1202
ChainResidue
ALEU1109
APRO1110
AARG1173
A2LL1201
AHOH1353

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1203
ChainResidue
ATYR1175
A2LL1201
AHOH1347

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

221716

PDB entries from 2024-06-26

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