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4NIE

Crystal structure of the orphan nuclear receptor ROR(gamma)t ligand-binding domain in complex with small molecule ligand

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE NBH A 601
ChainResidue
ACYS285
AALA368
APHE377
APHE378
ATYR502
AHOH735
AGLN286
ALEU287
ATRP317
ACYS320
AHIS323
AARG364
AMET365
AARG367

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE DMX A 602
ChainResidue
ATRP314
AHIS490
APRO491
AILE492
AVAL493
BGLU333

site_idAC3
Number of Residues17
DetailsBINDING SITE FOR RESIDUE NBH B 601
ChainResidue
BCYS285
BGLN286
BLEU287
BTRP317
BCYS320
BHIS323
BLEU324
BARG364
BMET365
BARG367
BALA368
BPHE377
BPHE378
BPHE388
BILE400
BTYR502
BHOH720

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE DMX B 602
ChainResidue
AGLU333
BTRP314
BLEU489
BHIS490
BPRO491
BILE492
BVAL493

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues478
DetailsDomain: {"description":"NR LBD","evidences":[{"source":"PROSITE-ProRule","id":"PRU01189","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues10
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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