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4N11

Crystal structure of plasmodium falciparum reduced glutaredoxin 1 (PfGrx1) complexed with cisplatin

Functional Information from GO Data
ChainGOidnamespacecontents
A0015038molecular_functionglutathione disulfide oxidoreductase activity
A0016209molecular_functionantioxidant activity
A0016491molecular_functionoxidoreductase activity
A0019153molecular_functionprotein-disulfide reductase (glutathione) activity
A0046872molecular_functionmetal ion binding
A0098869biological_processcellular oxidant detoxification
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE MPO A 201
ChainResidue
ASER5
AHOH302
AHOH327
AHOH362
ALYS9
ATYR31
ATYR65
AGLU68
APRO76
AGLY87
ACYS88
AASP89

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE MPD A 202
ChainResidue
AASN13
AGLU17
ALYS82
AHOH375

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE MPD A 203
ChainResidue
ALYS26
ATHR27
AGLU28
AILE33
AILE36
AHOH345

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CPT A 204
ChainResidue
ALYS26
AGLU28
ACYS29
AVAL75
AHOH377

Functional Information from PROSITE/UniProt
site_idPS00195
Number of Residues17
DetailsGLUTAREDOXIN_1 Glutaredoxin active site. VFakteCPYCikAisiL
ChainResidueDetails
AVAL23-LEU39

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PDB entries from 2024-10-09

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