4MGB
Crystal structure of hERa-LBD (Y537S) in complex with TCBPA
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 11 |
Details | BINDING SITE FOR RESIDUE XDH A 601 |
Chain | Residue |
A | LEU346 |
A | GLY521 |
A | LEU525 |
A | LEU349 |
A | ALA350 |
A | GLU353 |
A | LEU387 |
A | MET388 |
A | LEU391 |
A | ILE424 |
A | PHE425 |
site_id | AC2 |
Number of Residues | 12 |
Details | BINDING SITE FOR RESIDUE XDH B 601 |
Chain | Residue |
B | LEU346 |
B | LEU349 |
B | ALA350 |
B | GLU353 |
B | LEU387 |
B | MET388 |
B | PHE404 |
B | MET421 |
B | ILE424 |
B | PHE425 |
B | HIS524 |
B | LEU525 |
site_id | AC3 |
Number of Residues | 3 |
Details | BINDING SITE FOR RESIDUE GOL B 602 |
Chain | Residue |
B | GLU323 |
B | TRP393 |
B | GLY442 |
site_id | AC4 |
Number of Residues | 3 |
Details | BINDING SITE FOR RESIDUE GOL B 603 |
Chain | Residue |
B | GLN441 |
B | GLU444 |
B | ALA493 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | MOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163 |
Chain | Residue | Details |
C | SER698 | |
D | SER698 | |
B | HIS524 |
site_id | SWS_FT_FI2 |
Number of Residues | 1 |
Details | MOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106 |
Chain | Residue | Details |
B | SER537 |
site_id | SWS_FT_FI3 |
Number of Residues | 1 |
Details | LIPID: S-palmitoyl cysteine => ECO:0000250 |
Chain | Residue | Details |
B | CYS447 |