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4LUO

Fragment-Based Discovery of a Potent Inhibitor of Replication Protein A Protein-Protein Interactions

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0005634cellular_componentnucleus
A0006260biological_processDNA replication
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 1DZ A 201
ChainResidue
AARG31
AHOH393
AILE33
AARG43
ASER55
AMET57
ALEU87
AARG92
AVAL93
A1DZ202

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 1DZ A 202
ChainResidue
AARG7
AARG41
AMET57
AASN85
ALEU87
AVAL93
AILE95
A1DZ201
AHOH390
AHOH392

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsModified residue: {"description":"N-acetylmethionine","evidences":[{"source":"PubMed","id":"19413330","evidenceCode":"ECO:0007744"},{"source":"PubMed","id":"22223895","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues3
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"26474068","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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