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4LM3

Crystal structure of PDE10A2 with fragment ZT464

Functional Information from GO Data
ChainGOidnamespacecontents
A0004114molecular_function3',5'-cyclic-nucleotide phosphodiesterase activity
A0007165biological_processsignal transduction
A0008081molecular_functionphosphoric diester hydrolase activity
B0004114molecular_function3',5'-cyclic-nucleotide phosphodiesterase activity
B0007165biological_processsignal transduction
B0008081molecular_functionphosphoric diester hydrolase activity
Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE 9ZE A 801
ChainResidue
ATYR524
ASER677
AMET713
AGLN726
APHE729
AHOH946
BLEU706

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE NI A 802
ChainResidue
AASP564
AASP674
AHOH930
AHOH1025
AHIS529
AHIS563

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE NI A 803
ChainResidue
AASP564
AHOH1023
AHOH1024
AHOH1025
AHOH1026
AHOH1027

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 804
ChainResidue
AMET648
ASER660
AARG716
AASP717
ALYS718
ALYS719
AASP720

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 805
ChainResidue
ALYS686
AALA689
AASN690
ATYR693

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO B 801
ChainResidue
AGLN576
ATHR588
ASER589
AASP634
BGLN709
BPRO710
BHOH1068

site_idAC7
Number of Residues7
DetailsBINDING SITE FOR RESIDUE NI B 802
ChainResidue
BHIS529
BHIS563
BASP564
BASP674
BNI803
BHOH1010
BHOH1012

site_idAC8
Number of Residues7
DetailsBINDING SITE FOR RESIDUE NI B 803
ChainResidue
BASP564
BNI802
BHOH942
BHOH1011
BHOH1012
BHOH1013
BHOH1014

Functional Information from PROSITE/UniProt
site_idPS00126
Number of Residues12
DetailsPDEASE_I_1 3'5'-cyclic nucleotide phosphodiesterase domain signature. HDLdHrGfsNsY
ChainResidueDetails
AHIS563-TYR574

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:18477562, ECO:0007744|PDB:2ZMF
ChainResidueDetails
AASN572
ASER616
AGLN650
AMET669
BASN572
BSER616
BGLN650
BMET669

237735

PDB entries from 2025-06-18

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