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4KO0

CRYSTAL STRUCTURE OF HIV-1 REVERSE TRANSCRIPTASE (RT) IN COMPLEX WITH an anilinylpyrimidine derivative (JLJ-135)

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0003964molecular_functionRNA-directed DNA polymerase activity
A0004523molecular_functionRNA-DNA hybrid ribonuclease activity
A0006278biological_processRNA-templated DNA biosynthetic process
B0003964molecular_functionRNA-directed DNA polymerase activity
B0006278biological_processRNA-templated DNA biosynthetic process
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE JLJ A 601
ChainResidue
ALEU100
AHIS235
ATYR318
BGLU138
ALYS101
ALYS103
AVAL106
AVAL179
ATYR181
ATYR188
APHE227
ALEU234

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 602
ChainResidue
ALYS331
AGLN334
ALYS512
AHOH876

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 603
ChainResidue
ALYS476
ASER515
AGLU516
ALEU517

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 604
ChainResidue
ATRP426
ATYR427
AGLN509
AASP511
AHOH718

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 501
ChainResidue
BTRP24
BGLU399
BTRP402
BTHR403
BHOH623

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING:
ChainResidueDetails
BASP110
BASP185
BASP186

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Essential for RT p66/p51 heterodimerization
ChainResidueDetails
BTRP401
BTRP414
AASP498
AASP549

site_idSWS_FT_FI3
Number of Residues2
DetailsSITE: Essential for RT p66/p51 heterodimerization
ChainResidueDetails
ATRP401
ATRP414

site_idSWS_FT_FI4
Number of Residues1
DetailsSITE: Cleavage; by viral protease; partial
ChainResidueDetails
APHE440

222415

PDB entries from 2024-07-10

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