4JFI
Increasing the Efficiency Efficiency of Ligands for the FK506-Binding Protein 51 by Conformational Control: Complex of FKBP51 with compound 1-[(9S,13R,13aR)-1,3-dimethoxy-8-oxo-5,8,9,10,11,12,13,13a-octahydro-6H-9,13-epiminoazocino[2,1-a]isoquinolin-14-yl]-2-(3,4,5-trimethoxyphenyl)ethane-1,2-dione
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003755 | molecular_function | peptidyl-prolyl cis-trans isomerase activity |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 13 |
Details | BINDING SITE FOR RESIDUE 1KT A 201 |
Chain | Residue |
A | TYR57 |
A | TYR113 |
A | SER118 |
A | LYS121 |
A | PHE130 |
A | PHE67 |
A | ASP68 |
A | ARG73 |
A | PHE77 |
A | GLN85 |
A | VAL86 |
A | ILE87 |
A | TRP90 |
site_id | AC2 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE DMS A 202 |
Chain | Residue |
A | LYS38 |
A | THR46 |
A | ALA95 |
A | HOH354 |
site_id | AC3 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE GOL A 203 |
Chain | Residue |
A | ALA14 |
A | GLU44 |
A | LYS60 |
A | HIS104 |
A | GLU131 |
A | HOH324 |
A | HOH477 |
Functional Information from SwissProt/UniProt
Chain | Residue | Details |
A | LYS28 | |