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4IR6

Crystal Structure of the bromodomain of human BAZ2B in complex with 1-{1-[2-(METHYLSULFONYL)PHENYL]-7-PHENOXYINDOLIZIN-3-YL}ETHANONE (GSK2838097A)

Functional Information from PDB Data
site_idAC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2001
ChainResidue
AASP1938
AGLU1941
ATHR1942

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2002
ChainResidue
AHIS1883
AGLU1884
AHOH2181

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2003
ChainResidue
AARG1864
ATHR1968
AHOH2177

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 2004
ChainResidue
AMET1875
AGLU1879
ATHR1968
AHOH2247

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 2005
ChainResidue
ATHR1878
AGLU1881
AARG1915
AHOH2301

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2006
ChainResidue
AGLU1927
ATRP1965
ALYS1970

site_idAC7
Number of Residues12
DetailsBINDING SITE FOR RESIDUE IR6 A 2007
ChainResidue
ATRP1887
APRO1888
ALEU1891
APRO1892
AVAL1893
AASN1894
AVAL1898
APRO1899
AASN1944
AILE1950
AHOH2211
AHOH2256

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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