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4IR5

Crystal Structure of the bromodomain of human BAZ2B in complex with 1-{1-[2-(hydroxymethyl)phenyl]-7-phenoxyindolizin-3-yl}ethanone (GSK2847449A)

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 2001
ChainResidue
AGLY1900
AASN1944
AILE1950
AEDO2009
AIR52013
AHOH2119
AHOH2135

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 2002
ChainResidue
AHOH2341
AHOH2341
AIR52013
AIR52013

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2003
ChainResidue
AASP1938
AGLU1941
ATHR1942
AARG1958
AHOH2226

site_idAC4
Number of Residues1
DetailsBINDING SITE FOR RESIDUE EDO A 2004
ChainResidue
ALYS1863

site_idAC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2005
ChainResidue
AASP1947
AARG1952
AEDO2012

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 2006
ChainResidue
AIR52013
AHOH2316

site_idAC7
Number of Residues8
DetailsBINDING SITE FOR RESIDUE EDO A 2007
ChainResidue
ATRP1887
APRO1888
ALEU1890
ALEU1891
APRO1892
AIR52013
AHOH2158
AHOH2234

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2008
ChainResidue
AMET1875
AGLU1879
ATHR1968
AHOH2295
AHOH2334

site_idAC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 2009
ChainResidue
ALEU1895
ALYS1896
APRO1899
AGLY1900
AEDO2001
AHOH2268

site_idBC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 2010
ChainResidue
AVAL1904
AILE1905
ALYS1906
ATHR1942
AHOH2132
AHOH2215
AHOH2323

site_idBC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 2011
ChainResidue
AGLU1962
AHOH2232
AHOH2245
AHOH2300

site_idBC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2012
ChainResidue
AASP1946
AARG1952
AHIS1955
AASN1956
AEDO2005

site_idBC4
Number of Residues13
DetailsBINDING SITE FOR RESIDUE IR5 A 2013
ChainResidue
APRO1888
AVAL1893
AASN1894
ALEU1897
APRO1899
AASN1944
AILE1950
AEDO2001
AEDO2002
AEDO2002
AEDO2006
AEDO2007
AHOH2123

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

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PDB entries from 2025-12-17

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