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4IA2

Diastereotopic and Deuterium Effects in Gemini

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues17
DetailsBINDING SITE FOR RESIDUE BIV A 501
ChainResidue
ATYR175
ACYS316
AVAL328
AHIS333
ALEU337
ALEU338
ALEU341
ALEU419
AHIS423
ATYR179
ALEU261
AVAL262
ASER265
AARG302
ASER303
ASER306
ATRP314

site_idAC2
Number of Residues17
DetailsBINDING SITE FOR CHAIN B OF NUCLEAR RECEPTOR COACTIVATOR 2
ChainResidue
AILE270
ALYS274
AARG280
AALA284
AGLN287
AILE288
ALYS292
APRO434
AGLU435
AMET438
ALEU443
AGLU446
AVAL447
AHOH614
BHOH701
BHOH703
BHOH705

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues18
DetailsRegion: {"description":"Interaction with coactivator LXXLL motif","evidences":[{"source":"UniProtKB","id":"P13053","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"UniProtKB","id":"P11473","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"17218092","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2HC4","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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