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4HKN

Complex structure of human tankyrase 2 with luteolin

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1202
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1203
ChainResidue
AASN990
AARG991
CPRO1160
CGLU1161
CHOH1305

site_idAC4
Number of Residues9
DetailsBINDING SITE FOR RESIDUE LU2 A 1204
ChainResidue
AHIS1031
AGLY1032
ATYR1060
APHE1061
AALA1062
ASER1068
ATYR1071
AHOH1347
CGLU1138

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 C 1201
ChainResidue
CHIS1117
CSER1118
CTYR1142
CARG1143
CHOH1308

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092

224004

PDB entries from 2024-08-21

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