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4HKK

Complex structure of human tankyrase 2 with apigenin

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ ADP-ribosyltransferase activity
D0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1202
ChainResidue
AHOH1378
BHOH1310
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1203
ChainResidue
AASN990
AARG991
BPRO1160
BGLU1161
BHOH1302

site_idAC4
Number of Residues12
DetailsBINDING SITE FOR RESIDUE AGI A 1204
ChainResidue
AHIS1031
AGLY1032
ATYR1050
ATYR1060
APHE1061
AALA1062
ALYS1067
ASER1068
ATYR1071
AHOH1398
AHOH1401
BGLU1138

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE PEG B 1201
ChainResidue
ATRP1006
AARG1100
BTYR1148
BGLU1150

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN C 1201
ChainResidue
CCYS1081
CHIS1084
CCYS1089
CCYS1092

site_idAC7
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 C 1202
ChainResidue
CARG977
CHIS979
CARG980
CLYS1067
CGLN1070
CHOH1372
CHOH1395
DHOH1209

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 C 1203
ChainResidue
CASN990
CARG991
DPRO1160
DGLU1161
DHOH1206

site_idAC9
Number of Residues3
DetailsBINDING SITE FOR RESIDUE PEG C 1204
ChainResidue
CLYS999
CTRP1006
DTYR1148

site_idBC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE AGI C 1205
ChainResidue
CHIS1031
CGLY1032
CTYR1050
CTYR1060
CPHE1061
CALA1062
CSER1068
CTYR1071
CHOH1385
DGLU1138

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
CCYS1081
CHIS1084
CCYS1089
CCYS1092

224201

PDB entries from 2024-08-28

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