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4GPQ

Structural insights into inhibition of the bivalent menin-MLL interaction by small molecules in leukemia

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
Functional Information from PDB Data
site_idAC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE PEG A 601
ChainResidue
ATYR319
AHOH1115

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE PG4 A 602
ChainResidue
ALEU75
ATHR76
ATYR361
APHE365
AHOH718
AHOH912
AHOH935

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE PEG A 603
ChainResidue
ATRP126
ASER130
ALYS135
ATRP198

site_idAC4
Number of Residues10
DetailsBINDING SITE FOR RESIDUE EPE A 604
ChainResidue
AVAL50
AASN331
AARG332
AASN333
AVAL334
AARG335
AGLY401
AALA403
AHOH936
AHOH1218

246704

PDB entries from 2025-12-24

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