4FDN
Mycobacterium tuberculosis DprE1 in complex with CT325 - hexagonal crystal form
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003885 | molecular_function | D-arabinono-1,4-lactone oxidase activity |
A | 0005886 | cellular_component | plasma membrane |
A | 0016020 | cellular_component | membrane |
A | 0016491 | molecular_function | oxidoreductase activity |
A | 0035884 | biological_process | arabinan biosynthetic process |
A | 0042597 | cellular_component | periplasmic space |
A | 0045227 | biological_process | capsule polysaccharide biosynthetic process |
A | 0046677 | biological_process | response to antibiotic |
A | 0050660 | molecular_function | flavin adenine dinucleotide binding |
A | 0070592 | biological_process | cell wall polysaccharide biosynthetic process |
A | 0071555 | biological_process | cell wall organization |
A | 0071949 | molecular_function | FAD binding |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 34 |
Details | BINDING SITE FOR RESIDUE FAD A 900 |
Chain | Residue |
A | TRP16 |
A | TYR60 |
A | ASN63 |
A | ALA64 |
A | MET74 |
A | ALA94 |
A | PRO116 |
A | GLY117 |
A | THR118 |
A | VAL121 |
A | THR122 |
A | ILE52 |
A | GLY124 |
A | GLY125 |
A | ALA128 |
A | CYS129 |
A | ILE131 |
A | HIS132 |
A | ASN178 |
A | GLY179 |
A | GLY182 |
A | ILE184 |
A | ALA53 |
A | TYR415 |
A | ALA417 |
A | 0T4901 |
A | HOH1015 |
A | HOH1023 |
A | ARG54 |
A | GLY55 |
A | LEU56 |
A | GLY57 |
A | ARG58 |
A | SER59 |
site_id | AC2 |
Number of Residues | 9 |
Details | BINDING SITE FOR RESIDUE 0T4 A 901 |
Chain | Residue |
A | TYR60 |
A | GLY117 |
A | GLY133 |
A | LYS134 |
A | VAL365 |
A | LYS367 |
A | ASN385 |
A | CYS387 |
A | FAD900 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | BINDING: BINDING => ECO:0000269|PubMed:22733761, ECO:0000269|PubMed:23776209, ECO:0000269|PubMed:24500695, ECO:0000269|PubMed:25427196, ECO:0007744|PDB:4FDP, ECO:0007744|PDB:4NCR |
Chain | Residue | Details |
A | ALA53 |
site_id | SWS_FT_FI2 |
Number of Residues | 5 |
Details | BINDING: BINDING => ECO:0000269|PubMed:22733761, ECO:0000269|PubMed:23776209, ECO:0000269|PubMed:24500695, ECO:0000269|PubMed:25427196, ECO:0007744|PDB:4FDP, ECO:0007744|PDB:4KW5, ECO:0007744|PDB:4NCR |
Chain | Residue | Details |
A | GLY117 | |
A | THR122 | |
A | CYS129 | |
A | ILE184 | |
A | TYR415 |