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4F1L

Human Artd8 (Parp14, Bal2) - catalytic domain in complex with inhibitor A16(Z)

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ ADP-ribosyltransferase activity
D0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE 0RY A 1801
ChainResidue
AHIS1601
ALEU1701
AHOH1925
AHOH1945
BTYR1646
B0RY1801
AGLY1602
AASN1624
ATYR1633
APHE1634
AALA1635
ATYR1640
ASER1641
ATYR1646

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE NO3 A 1802
ChainResidue
APHE1536
APRO1609
AASN1612
AARG1613
DPHE1536
DVAL1608
DPRO1609
DASN1612

site_idAC3
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 0RY B 1801
ChainResidue
AVAL1626
AASN1643
ATYR1646
A0RY1801
BHIS1601
BGLY1602
BTYR1633
BPHE1634
BALA1635
BSER1641
BTYR1646
BLEU1701
BHOH1969

site_idAC4
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 0RY C 1801
ChainResidue
CHIS1601
CGLY1602
CASN1624
CVAL1626
CTYR1633
CPHE1634
CALA1635
CTYR1640
CSER1641
CTYR1646
CLEU1701
CHOH1937
DTYR1646

site_idAC5
Number of Residues8
DetailsBINDING SITE FOR RESIDUE NO3 C 1802
ChainResidue
BPHE1536
BVAL1608
BPRO1609
BASN1612
CPHE1536
CPRO1609
CASN1612
CARG1613

site_idAC6
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 0RY D 1801
ChainResidue
CASN1643
CTHR1645
CTYR1646
DHIS1601
DGLY1602
DVAL1626
DTYR1633
DALA1635
DTYR1640
DSER1641
DTYR1646

221716

PDB entries from 2024-06-26

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