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4E0O

SVQIVYK segment from human Tau (305-311) displayed on 54-membered macrocycle scaffold (form III)

Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE MPD A 101
ChainResidue
AVAL5
AGLU9
APHE10
AHAO11

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MPD A 102
ChainResidue
AVAL2
AHAO11
A4BF12
BHAO11
B4BF12

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PO4 B 101
ChainResidue
BTYR6
BORN8
BHOH203
BHOH209
BHOH212
BHOH213

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MPD B 102
ChainResidue
BVAL5
BGLU9
BPHE10
BHAO11
BHOH216

site_idAC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE MPD B 103
ChainResidue
BGLN3
BVAL5
BHAO11

site_idAC6
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MPD C 101
ChainResidue
CGLN3
CVAL5
CHAO11
C4BF12
D4BF12

site_idAC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PO4 D 101
ChainResidue
DTYR6
DORN8
DPO4102
DHOH207
DHOH209
DHOH210

site_idAC8
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PO4 D 102
ChainResidue
DORN8
DPO4101
DHOH201
DHOH208
DHOH211
DHOH212

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MPD D 103
ChainResidue
CVAL2
CHAO11
C4BF12
DHAO11
D4BF12

site_idBC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE MPD D 104
ChainResidue
DVAL5
DGLU9
DPHE10
DHAO11

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsSITE: Not glycated => ECO:0000269|PubMed:9326300
ChainResidueDetails
ALYS7
BLYS7
CLYS7
DLYS7

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine; by PHK => ECO:0000269|PubMed:7706316, ECO:0000269|PubMed:8999860
ChainResidueDetails
ASER1
BSER1
CSER1
DSER1

site_idSWS_FT_FI3
Number of Residues4
DetailsMOD_RES: N6-acetyllysine; alternate => ECO:0000250|UniProtKB:P10637
ChainResidueDetails
ALYS7
BLYS7
CLYS7
DLYS7

site_idSWS_FT_FI4
Number of Residues8
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin); in PHF-tau => ECO:0000269|PubMed:16443603
ChainResidueDetails
ALYS7
BLYS7
CLYS7
DLYS7

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PDB entries from 2024-07-24

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